Description
SR-14968 is an opioid analgesic drug, an derivative of brorphine and SR-17018, acting as an agonist of the μ-opioid receptor. This drug exhibits agonistic agonist activity in vitro at higher dosages, as shown by in vivo mouse studies, and has a higher safety profile compared to fentanyl.
This preparation is a research drug designed for scientific purposes, as well as to identify analgesic drug with a lower risk of overdose compared to traditional opioids.
Chemistry
SR-17018 is closely related to compounds such as brorphine and SR-17018.
Pharmacology, Pharmacodynamic
Studies in mice have shown that SR-14968 acts as an agonist of the μ-opioid receptor, which is selective for activating the G-protein signaling pathway over β-arrestin 2 recruitment, which is responsible for the analgesic effect. This drug can also cause relaxing and hypnotic effects.
Toxicological and pharmacological properties in the process of studying on rodents in laboratory conditions.
Dosage
The exact dosages of the drug have not been established. In the process of studying.
Legal status
It is not controlled in many countries at the moment.
Technical Information:
Product Name SR-14968
Synonyms US10751335, Example 2
IUPAC Name 3-[1-[1-(4-bromophenyl)ethyl]piperidin-4-yl]-5,6-dichloro-1H-benzimidazol-2-one
CAS Number 2133455-40-8
Molecular Formula C20H20BrCl2N3O
Formula Weight 469.2 g/mol
InChi Code InChI=1S/C20H20BrCl2N3O/c1-12(13-2-4-14(21)5-3-13)25-8-6-15(7-9-25)26-19-11-17(23)16(22)10-18(19)24-20(26)27/h2-5,10-12,15H,6-9H2,1H3,(H,24,27)
InChi Key DJSSLECNUQMYKG-UHFFFAOYSA-N
SMILES CC(C1=CC=C(C=C1)Br)N2CCC(CC2)N3C4=CC(=C(C=C4NC3=O)Cl)Cl
Solubility
Acetone: Soluble
DMSO: Soluble
Formulation A solid
Purity ≥98%
Disclaimer of liability
DPP-26 is intended only as a substance for scientific and research purposes in special laboratory conditions in compliance with all standards and safety measures.
You can buy DPP-26 online at ChemicalNS company right now and participate in our bonus program, or you can become our partners.
Why is it worth buying SR-14968 online at ChemicalNS company?
-We are a chemical company that has proven itself in the chemical industry market, which is ready to share its experience in scientific circles and ready to supply innovative chemical products in the scientific environment, for research and tests.
-All ChemicalNS company products have been tested and verified.
-Product purity 98-99%.
-You will receive a ZIP Pack, a sealed aluminum foil package containing the research product.
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