Description
SR-17018 is an opioid drug acting as a biased agonist of the μ-opioid receptor, by activating a signaling G protein on top of the recruitment of β-arrestin, acting as an analgesic with the least respiratory depression unlike other opioid drugs. This substance is relatively new and is positioned as a research drug for chemical and scientific research, to identify pharmacological, analgesic features.
Pharmacology, Pharmacodynamics
Studies have shown that SR-17018 acts as a mixed agonist of the μ-opioid receptor and causes effects such as analgesia, sedation, relaxation, and euphoria. SR-17018, unlike heroin and morphine, causes fewer side effects such as itching, respiratory depression and the development of tolerance.
Toxicological and pharmacological properties in the process of studying rodents in the laboratory.
Side effects
With improper use, high dosage, as well as use with other drugs, side effects such as respiratory depression, delirium, nausea, itching and constipation, physical and psychological addiction are possible.
Dosage
The exact dosage is not known, due to the lack of proper medical research. It has been established that SR-17018 is a potent analgesic with high opioid activity, therefore it is necessary to be extremely careful with dosages.
Legal status
The legal status is not clear. It is legal in many countries as a means for research and scientific work.
Technical Information:
Product Name SR-17018
Synonyms SR17018
IUPAC Name 5,6-dichloro-3-[1-[(4-chlorophenyl)methyl]piperidin-4-yl]-1H-benzimidazol-2-one
CAS Number 2134602-45-0
Molecular Formula C19H18Cl3N3O
Formula Weight 410.72 g·mol−1
InChi Code InChI=1S/C19H18Cl3N3O/c20-13-3-1-12(2-4-13)11-24-7-5-14(6-8-24)25-18-10-16(22)15(21)9-17(18)23-19(25)26/h1-4,9-10,14H,5-8,11H2,(H,23,26)
InChi Key LAGUDYUGRSQDKS-UHFFFAOYSA-N
SMILES C1CN(CCC1N2C3=CC(=C(C=C3NC2=O)Cl)Cl)CC4=CC=C(C=C4)Cl
Solubility
DMF: 1 mg/ml
DMSO: 1 mg/ml
DMSO:PBS (pH 7.2) (1:2): 0.33 mg/ml
Ethanol: slightly soluble
Formulation A crystalline solid
Purity ≥98%
Disclaimer of liability
SR-17018 is intended only as a substance for scientific and research purposes in special laboratory conditions in compliance with all standards and safety measures.
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-Product purity 98-99%.
-You will receive a ZIP Pack, a sealed aluminum foil package containing the research product.
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